吐根酚碱盐酸盐 EP

中文名	吐根酚碱盐酸盐 EP
英文名	Cephaeline hydrochloride
别名	盐酸吐根酚碱吐根酚碱盐酸盐 EP 吐根酚碱盐酸盐 EP标准品吐根酚碱盐酸盐(盐酸吐根酚碱)
英文别名	NSC 32944 Cephaeline DiHCl Cephaeline HCl salt cephaelin hydrochloride Cephaeline hydrochloride cephaeline hydrochloride Cephaeline dihydrochloride Cephaeline hydrochloride CRS (-)-CEPHAELINE DIHYDROCHLORIDE (1R)-1-[[(2S,3R,11bS)-3-Ethyl-1,3,4,6,7,11b-hexahydro-9,10-dimethoxy-2H-benzo[a]quinolizin-2-yl]methyl]-1,2,3,4-tetrahydro-7-methoxy-6-isoquinolinol hydrochloride
CAS	5853-29-2
EINECS	227-463-3
化学式	C28H39ClN2O4
分子量	503.08
存储条件	2-8℃
外观	整洁
物化性质	类白至黄色粉末，可溶于甲醇、乙醇、DMSO等有机溶剂，来源于吐根，安哥拉八角枫。
体外研究	CYP2D6 reveals the highest metabolic activity for the generation of 9-O-demethylEmetine, whereas this enzyme also shows a significant metabolic activity for the generation of Cephaeline. The IC 50 s of Cephaeline against CYP2C9, CYP2D6 and CYP3A4 is over 1000, 121 and 1000 μM, respectively. Further experiments are performed to determine inhibition constants (K i ) for Cephaeline on the CYP2D6 and CYP3A4 activities Graphic analysis of Dixon plots at various Cephaeline concentrations for each of the two CYP enzyme assays yield K i s of 54 and 355 μM for CYP2D6 and CYP3A4, respectively.
危险品运输编号	1544
Hazard Class	6.1(b)
Packing Group	III

吐根酚碱盐酸盐 EP - 配置溶液浓度参考

	1mg	5mg	10mg
1 mM	1.853 ml	9.267 ml	18.534 ml
5 mM	0.371 ml	1.853 ml	3.707 ml
10 mM	0.185 ml	0.927 ml	1.853 ml
5 mM	0.037 ml	0.185 ml	0.371 ml

最后更新：2024-01-02 23:10:35

湖北扬信医药科技有限公司

产品名: 吐根碱双盐酸盐询盘
CAS: 5853-29-2
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产品名: 盐酸吐根酚碱去供应商网站查看询盘
CAS: 5853-29-2
产地: 上海
规格: C889731
价格: 20mg-1794
库存: 7天内发货
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